Relebactam | ||||
CAS NO.: | 1174018-99-5 | |||
Chemical Formula: | C12H20N4O6S | |||
Molecular Weight: | 348.3800 | |||
DMF&GMP status: | Please contact us for more details. | Description: |
Relebactam is a diazabicyclooctane beta-lactamase inhibitor, similar in structure to [avibactam]. It includes a piperidine ring which reduces export from bacterial cells by producing a positive charge. It is currently available in a combination product which includes [imipenem] and [cilastatin] to treat complicated urinary tract infections (UTIs), pyelonephritis, and complicated intra-abdominal infections in adults. It is considered to be a last-line treatment option and gained FDA approval as part of the combination product RecarbrioⓇ in July 2019.
**The products protected by patents in this product catalog are used for laboratory analysis, research and development, and cannot be sold to any country or region with patent protection and for commercial purpose. If the resulting patent infringement risks and responsibilities will be borne by the buyer. |
|
Approvals | ||||
Active Ingredient | Dosage Form; Route | Strength | Proprietary Name | Applicant |
CILASTATIN SODIUM; IMIPENEM; RELEBACTAM | POWDER;INTRAVENOUS | EQ 500MG BASE/VIAL; 500MG/VIAL; 250MG/VIAL | RECARBRIO | MERCK SHARP AND DOHME CORP A SUB OF MERCK AND CO INC |
Patent Data | ||||
Patent No. | Patent Expiration | Drug Substance Claim | Drug Product Claim | Patent Use Code |
8487093 | 11/19/2029 | DS | DP | U-2586 U-2587 U-2840 |
Exclusive Data | ||||
Exclusivity Code | Exclusivity Expiration | |||
N.A. | N.A. | |||